Name: RIGHTEOUS GSK-2881078
Brand: RIGHTEOUS SPORTS NUTRITION
SKU: HGMHFHZAHNHS6
Price: 79.95 USD
Availability: InStock

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RIGHTEOUS GSK-2881078

Product Details

Brand: RIGHTEOUS SPORTS NUTRITION

GSK-2881078 is a nonsteroidal selective androgen receptor modulator

Purpose: Developed by GlaxoSmithKline (GSK) for the treatment of reduced mobility and muscle weakness associated with chronic and acute illnesses. It was specifically explored for its potential to prevent muscle wasting and sarcopenia in older individuals.

Mechanism: As a SARM, GSK-2881078 binds to the androgen receptor, influencing its activity in a tissue-selective manner. This allows it to act as an agonist (activator) in tissues like muscle and bone, while potentially acting as an antagonist or partial agonist in other tissues like the prostate or skin. This selectivity aims to provide beneficial effects of androgen therapy without the undesirable side effects.

Clinical Trials:

A first-in-human study in 2017 investigated its safety, pharmacokinetics, and pharmacodynamics in healthy males and females.
A phase 1b study showed that GSK-2881078 was well-tolerated and produced dose-dependent increases in lean body mass in healthy older males and postmenopausal females.
A phase II trial demonstrated it was well tolerated and increased muscle strength in men with Chronic Obstructive Pulmonary Disease (COPD).

Research Focus: GSK-2881078 is evaluated for its effects on muscle growth and strength to improve physical function in individuals with muscle wasting.

In summary, GSK-2881078 is a selective androgen receptor modulator studied for its ability to improve muscle mass and strength, especially in people suffering from muscle wasting conditions

WARNING:

THIS IS NOT A DIETARY SUPPLEMENT. FOR RESEARCH PURPOSES ONLY!

NOT RESPONSIBLE FOR INJURIES.

ALL RESEARCHERS REPRESENT AND WARRANT THAT THROUGH THEIR OWN REVIEW AND STUDY, THEY ARE FULLY AWARE

AND KNOWLEDGEABLE ABOUT THE FOLLOWING PRODUCT.

ALL RESEARCHERS MUST BE 18 YEARS OR OLDER TO PURCHASE.

UNDER NO CIRCUMSTANCES SHALL RIGHTEOUS SPORTS NUTRITION BE LIABLE FOR CONSEQUENTIAL DAMAGES WHETHER PURCHASES

CLAIM CONTACT, NEGLIGENCE, STRICT LIABILITY OR OTHERWISE. IN PURCHASING THIS PRODUCT, PURCHASER AGREES TO THE ABOVE.